Compile Data Set for Download or QSAR
Found 17 of ic50 data for polymerid = 6211
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human MEK3 using p38alpha as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5KB8PubMed
LigandPNGBDBM50134589(CHEMBL3747095)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of MKK3 (unknown origin) using [gamma-33P]-ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7BXVPubMed
LigandPNGBDBM50134587(CHEMBL3746157)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of MKK3 (unknown origin) using [gamma-33P]-ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7BXVPubMed
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 17.2nMAssay Description:Inhibition of human MEK3 using p38alpha as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W380MTPubMed
LigandPNGBDBM50134590(CHEMBL3747443)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of MKK3 (unknown origin) using [gamma-33P]-ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7BXVPubMed
LigandPNGBDBM50134588(CHEMBL3746484)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of MKK3 (unknown origin) using [gamma-33P]-ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7BXVPubMed
LigandPNGBDBM103302(SCH772984 | US8546404, 6)copy SMILEScopy InChI
Affinity DataIC50: 304nMAssay Description:The IC50 values of selected kinases were determined using either Z'LYTE, Adapta or LanthaScreen assays.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8JCHPubMed
LigandPNGBDBM50141410((Z)-3-Amino-3-(2-amino-phenylsulfanyl)-2-[3-(hydro...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory potency against MAP kinase kinase 3 (MKK3)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H131F0PubMed
LigandPNGBDBM50375668(CHEMBL259526)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of MKK3Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB82RHPubMed
LigandPNGBDBM50134591(CHEMBL3745744)copy SMILEScopy InChI
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of MKK3 (unknown origin) using [gamma-33P]-ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7BXVPubMed
LigandPNGBDBM50235816(CHEMBL4069365)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MAP2K3 (unknown origin) after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ061VPubMed
LigandPNGBDBM50135286(CHEMBL3745885)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human MEK3 using p38alpha as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7WT8PubMed
LigandPNGBDBM50115298(4-(6,7-Dimethoxy-quinazolin-4-yl)-piperazine-1-car...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of MKK-3, Mitogen activated protein kinase kinase 3More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RX9BDPPubMed
LigandPNGBDBM50118831(4-(6,7-Dimethoxy-quinazolin-4-yl)-piperazine-1-car...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Mitogen activated protein kinase kinase 3More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JH3MXFPubMed
LigandPNGBDBM50115297(4-(6,7-Dimethoxy-quinazolin-4-yl)-piperazine-1-car...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of MKK-3, Mitogen activated protein kinase kinase 3More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RX9BDPPubMed
LigandPNGBDBM50115295(4-(6,7-Dimethoxy-quinazolin-4-yl)-piperazine-1-car...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of MKK-3, Mitogen activated protein kinase kinase 3More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RX9BDPPubMed
LigandPNGBDBM50097398(CHEMBL449216 | HTS-9026)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of MKK3 (unknown origin) using [gamma-33P]-ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7BXVPubMed